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5EDI
CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c2(c(n1nc(nc1c(c2)C)CCc3nc(nn3C)N4CCCC4)C)Cl, micromolar IC50=0.000279
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RCSB PDB Mol* Viewer 2.11.2 [1/27/2025, 4:56:27 PM]
Sequence of
TSEEWQGLMQ462 FTLPVRLCRE472 IELFHFDIGP482 FENMWPGIFV492 YMVHRSCGTS502 CFELEKLCMERF512 IMSVKKNYRR522 VPYHNWKHAV532 TVAHCMYAIL542 QNNHTLFTDL552 ERKGLLIACL562 CHDLDHRGFS572 NSYLQKFDHP582 LAALYSTSTM592 EQHHFSQTVS602 ILQLEGHNIF612 STLSSSEYEQ622 VLEIIRKAII632 ATDLALYFGN642 RKQLEEMYQT652 GSLNLNNQSH662 RDRVIGLMMT672 ACDLCSVTKL682 WPVTKLTAND692 IYAEFWAEGD702 EMKKLGIQPI712 PMMDRDKKDE722 VPQGQLGFYN732 AVAIPCYTTL742 TQILPPTEPL752 LKACRDNLSQ762 WEKVIRGEE
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Dynamic Bonds
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