Crystal Structure of a G12C Oncogenic Variant of Human KRas Bound to a Novel GDP Competitive Covalent Inhibitor

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RCSB PDB Mol* Viewer 2.11.2 [1/27/2025, 4:56:27 PM]
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0    ​G​​M​​T​​E​​Y​​K​​L​​V​​V​​V​10   ​G​​A​​C​​G​​V​​G​​K​​S​​A​​L​20   ​T​​I​​Q​​L​​I​​Q​​N​​H​​F​​V​30   ​D​​E​​Y​​D​​P​​T​​I​​E​​D​​S​40   ​Y​​R​​K​​Q​​V​​V​​I​​D​​G​​E​50   ​T​​C​​L​​L​​D​​I​​L​​D​​T​​A​60   ​G​​Q​​E​​E​​Y​​S​​A​​M​​R​​D​70   ​Q​​Y​​M​​R​​T​​G​​E​​G​​F​​L​80   ​C​​V​​F​​A​​I​​N​​N​​T​​K​​S​90   ​F​​E​​D​​I​​H​​H​​Y​​R​​E​​Q​100  ​I​​K​​R​​V​​K​​D​​S​​E​​D​​V​110  ​P​​M​​V​​L​​V​​G​​N​​K​​C​​D​120  ​L​​P​​S​​R​​T​​V​​D​​T​​K​​Q​130  ​A​​Q​​D​​L​​A​​R​​S​​Y​​G​​I​140  ​P​​F​​I​​E​​T​​S​​A​​K​​T​​R​150  ​Q​​G​​V​​D​​D​​A​​F​​Y​​T​​L​160  ​V​​R​​E​​I​​R​​K​​H​​K​​E​​K​
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