Crystal structure of the complex between PPARgamma and the partial agonist LT127 (ureidofibrate derivative). Structure obtained from crystals of the apo-form soaked for 30 days.

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RCSB PDB Mol* Viewer 2.11.2 [1/27/2025, 4:56:27 PM]
Sequence of
     ​G​​S​​H​​M​​A​​E​​I​​S​​S​​D​     ​I​​D​​Q​​L​​N​​P​​E​​S​​A​​D​211  ​L​​R​​A​​L​​A​​K​​H​​L​​Y​​D​221  ​S​​Y​​I​​K​​S​​F​​P​​L​​T​​K​231  ​A​​K​​A​​R​​A​​I​​L​​T​​G​​K​241  ​T​​T​​D​​K​​S​​P​​F​​V​​I​​Y​251  ​D​​M​​N​​S​​L​​M​​M​​G​​E​​D​261  ​K​​I​​K​​F​​K​​H​​I​​T​​P​​L​271  ​Q​​E​​Q​​S​​K​​E​​V​​A​​I​​R​281  ​I​​F​​Q​​G​​C​​Q​​F​​R​​S​​V​291  ​E​​A​​V​​Q​​E​​I​​T​​E​​Y​​A​301  ​K​​S​​I​​P​​G​​F​​V​​N​​L​​D​311  ​L​​N​​D​​Q​​V​​T​​L​​L​​K​​Y​321  ​G​​V​​H​​E​​I​​I​​Y​​T​​M​​L​331  ​A​​S​​L​​M​​N​​K​​D​​G​​V​​L​341  ​I​​S​​E​​G​​Q​​G​​F​​M​​T​​R​351  ​E​​F​​L​​K​​S​​L​​R​​K​​P​​F​361  ​G​​D​​F​​M​​E​​P​​K​​F​​E​​F​371  ​A​​V​​K​​F​​N​​A​​L​​E​​L​​D​381  ​D​​S​​D​​L​​A​​I​​F​​I​​A​​V​391  ​I​​I​​L​​S​​G​​D​​R​​P​​G​​L​401  ​L​​N​​V​​K​​P​​I​​E​​D​​I​​Q​411  ​D​​N​​L​​L​​Q​​A​​L​​E​​L​​Q​421  ​L​​K​​L​​N​​H​​P​​E​​S​​S​​Q​431  ​L​​F​​A​​K​​L​​L​​Q​​K​​M​​T​441  ​D​​L​​R​​Q​​I​​V​​T​​E​​H​​V​451  ​Q​​L​​L​​Q​​V​​I​​K​​K​​T​​E​461  ​T​​D​​M​​S​​L​​H​​P​​L​​L​​Q​471  ​E​​I​​Y​​K​​D​​L​
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