Structure Determination MethodologyScientific Name of Source OrganismRefinement Resolution (Å)Enzyme Classification Name | Wilbur, J.D., Hwang, P.K., Ybe, J.A., Lane, M., Sellers, B.D., Jacobson, M.P., Fletterick, R.J., Brodsky, F.M. (2010) Dev Cell 18: 841-848 Released | 2010-06-09 | Method | X-RAY DIFFRACTION 7.94 Å | Organisms | | Macromolecule | |
Wilbur, J.D., Hwang, P.K., Ybe, J.A., Lane, M., Sellers, B.D., Jacobson, M.P., Fletterick, R.J., Brodsky, F.M. (2010) Dev Cell 18: 841-848 Released | 2010-06-09 | Method | X-RAY DIFFRACTION 9 Å | Organisms | | Macromolecule | |
Vetting, M.W., Toro, R., Bhosle, R., Al Obaidi, N.F., Morisco, L.L., Wasserman, S.R., Sojitra, S., Zhao, S., Stead, M., Washington, E., Scott Glenn, A., Chowdhury, S., Evans, B., Hammonds, J., Hillerich, B., Love, J., Seidel, R.D., Imker, H.J., Jacobson, M.P., Gerlt, J.A., Almo, S.C., Enzyme Function Initiative (EFI) (2015) Biochemistry 54: 909-931 Released | 2013-09-04 | Method | X-RAY DIFFRACTION 1.6 Å | Organisms | | Macromolecule | | Unique Ligands | EPE, MLI |
Vetting, M.W., Toro, R., Bhosle, R., Al Obaidi, N.F., Zhao, S., Stead, M., Washington, E., Scott Glenn, A., Chowdhury, S., Evans, B., Hammonds, J., Hillerich, B., Love, J., Seidel, R.D., Imker, H.J., Jacobson, M.P., Gerlt, J.A., Almo, S.C., Enzyme Function Initiative (EFI) (2015) Biochemistry 54: 909-931 Released | 2013-09-04 | Method | X-RAY DIFFRACTION 1.8 Å | Organisms | | Macromolecule | | Unique Ligands | CIT, MLI |
Vetting, M.W., Toro, R., Bhosle, R., Al Obaidi, N.F., Morisco, L.L., Wasserman, S.R., Sojitra, S., Zhao, S., Stead, M., Washington, E., Scott Glenn, A., Chowdhury, S., Evans, B., Hammonds, J., Hillerich, B., Love, J., Seidel, R.D., Imker, H.J., Jacobson, M.P., Gerlt, J.A., Almo, S.C., Enzyme Function Initiative (EFI) (2015) Biochemistry 54: 909-931 Released | 2013-09-18 | Method | X-RAY DIFFRACTION 1.46 Å | Organisms | | Macromolecule | | Unique Ligands | BDP, GCU |
Vetting, M.W., Toro, R., Bhosle, R., Al Obaidi, N.F., Morisco, L.L., Wasserman, S.R., Sojitra, S., Zhao, S., Stead, M., Washington, E., Scott Glenn, A., Chowdhury, S., Evans, B., Hammonds, J., Hillerich, B., Love, J., Seidel, R.D., Imker, H.J., Jacobson, M.P., Gerlt, J.A., Almo, S.C., Enzyme Function Initiative (EFI) (2015) Biochemistry 54: 909-931 Released | 2013-09-18 | Method | X-RAY DIFFRACTION 1.1 Å | Organisms | | Macromolecule | | Unique Ligands | ADA, CL, EDO, GTR |
Vetting, M.W., Toro, R., Bhosle, R., Al Obaidi, N.F., Morisco, L.L., Wasserman, S.R., Sojitra, S., Zhao, S., Stead, M., Scott Glenn, A., Chowdhury, S., Evans, B., Hillerich, B., Love, J., Seidel, R.D., Imker, H.J., Jacobson, M.P., Gerlt, J.A., Almo, S.C., Enzyme Function Initiative (EFI) (2015) Biochemistry 54: 909-931 Released | 2013-09-25 | Method | X-RAY DIFFRACTION 1.05 Å | Organisms | | Macromolecule | | Unique Ligands | 173, SO4 |
Vetting, M.W., Toro, R., Bhosle, R., Al Obaidi, N.F., Morisco, L.L., Wasserman, S.R., Sojitra, S., Zhao, S., Stead, M., Scott Glenn, A., Chowdhury, S., Evans, B., Hillerich, B., Love, J., Seidel, R.D., Imker, H.J., Jacobson, M.P., Gerlt, J.A., Almo, S.C., Enzyme Function Initiative (EFI) (2015) Biochemistry 54: 909-931 Released | 2013-09-25 | Method | X-RAY DIFFRACTION 1.9 Å | Organisms | | Macromolecule | | Unique Ligands | 173 |
Vetting, M.W., Toro, R., Bhosle, R., Al Obaidi, N.F., Morisco, L.L., Wasserman, S.R., Sojitra, S., Zhao, S., Stead, M., Attonito, J.D., Scott Glenn, A., Chowdhury, S., Evans, B., Hillerich, B., Love, J., Seidel, R.D., Imker, H.J., Jacobson, M.P., Gerlt, J.A., Almo, S.C., Enzyme Function Initiative (EFI) (2015) Biochemistry 54: 909-931 Released | 2013-10-16 | Method | X-RAY DIFFRACTION 1.1 Å | Organisms | | Macromolecule | | Unique Ligands | CL, SIN |
Kim, J., Toro, R., Bhosle, R., Al Obaidi, N.F., Morisco, L.L., Wasserman, S.R., Sojitra, S., Washington, E., Glenn, A.S., Chowdhury, S., Evans, B., Zhao, S.C., Hillerich, B., Love, J., Seidel, R.D., Imker, H.J., Stead, M., Jacobson, M.P., Gerlt, J.A., Almo, S.C., Enzyme Function Initiative (EFI) To be published Released | 2013-10-16 | Method | X-RAY DIFFRACTION 1.7 Å | Organisms | | Macromolecule | |
Vetting, M.W., Toro, R., Bhosle, R., Al Obaidi, N.F., Zhao, S., Stead, M., Attonito, J.D., Scott Glenn, A., Chowdhury, S., Evans, B., Hillerich, B., Love, J., Seidel, R.D., Imker, H.J., Jacobson, M.P., Gerlt, J.A., Almo, S.C., Enzyme Function Initiative (EFI) (2015) Biochemistry 54: 909-931 Released | 2013-10-16 | Method | X-RAY DIFFRACTION 1.651 Å | Organisms | | Macromolecule | | Unique Ligands | BDP, MG |
Vetting, M.W., Toro, R., Bhosle, R., Al Obaidi, N.F., Zhao, S., Stead, M., Attonito, J.D., Scott Glenn, A., Chowdhury, S., Evans, B., Hillerich, B., Love, J., Seidel, R.D., Imker, H.J., Jacobson, M.P., Gerlt, J.A., Almo, S.C., Enzyme Function Initiative (EFI) (2015) Biochemistry 54: 909-931 Released | 2013-10-16 | Method | X-RAY DIFFRACTION 1.501 Å | Organisms | | Macromolecule | | Unique Ligands | CA, CL, GTR |
Patskovsky, Y., Vetting, M.W., Toro, R., Bhosle, R., Al Obaidi, N., Stead, M., Washington, E., Scott Glenn, A., Chowdhury, S., Evans, B., Hammonds, J., Hillerich, B., Love, J., Seidel, R.D., Imker, H.J., Jacobson, M.P., Gerlt, J.A., Almo, S.C., Enzyme Function Initiative (EFI) (2015) Biochemistry 54: 909-931 Released | 2013-10-23 | Method | X-RAY DIFFRACTION 1.57 Å | Organisms | | Macromolecule | | Unique Ligands | GOL |
Kim, J., Toro, R., Bhosle, R., Al Obaidi, N.F., Morisco, L.L., Wasserman, S.R., Sojitra, S., Washington, E., Glenn, A.S., Chowdhury, S., Evans, B., Zhao, S.C., Hillerich, B., Love, J., Seidel, R.D., Imker, H.J., Stead, M., Jacobson, M.P., Gerlt, J.A., Almo, S.C., Enzyme Function Initiative (EFI) To be published Released | 2013-11-06 | Method | X-RAY DIFFRACTION 2.69 Å | Organisms | | Macromolecule | |
Bruning, J.M., Wang, Y., Otrabella, F., Boxue, T., Liu, H., Bhattacharya, P., Guo, S., Holton, J.M., Fletterick, R.J., Jacobson, M.P., England, P.M. (2019) Cell Chem Biol 26: 674-685.e6 Released | 2019-03-20 | Method | X-RAY DIFFRACTION 3.2 Å | Organisms | | Macromolecule | | Unique Ligands | BR, G7J, K |
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