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6EIX
Crystal structure of the kinase domain of the Q207E mutant of ACVR1 (ALK2) in complex with a 2-aminopyridine inhibitor K02288
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RCSB PDB Mol* Viewer 2.11.2 [1/27/2025, 4:56:27 PM]
Sequence of
SMTTNVGDST LADLLDHSCT SGSGSGLPFL200 VQRTVAREIT210 LLECVGKGRY220 GEVWRGSWQG230 ENVAVKIFSS240 RDEKSWFRET250 ELYNTVMLRH260 ENILGFIASD270 MTSRHSSTQL280 WLITHYHEMG290 SLYDYLQLTT300 LDTVSCLRIV310 LSIASGLAHL320 HIEIFGTQGK330 PAIAHRDLKS340 KNILVKKNGQ350 CCIADLGLAV360 MHSQSTNQLD370 VGNNPRVGTK380 RYMAPEVLDE390 TIQVDCFDSY400 KRVDIWAFGL410 VLWEVARRMV420 SNGIVEDYKP430 PFYDVVPNDP440 SFEDMRKVVC450 VDQQRPNIPN460 RWFSDPTLTS470 LAKLMKECWY480 QNPSARLTAL490 RIKKTLTKID500 NSLDKLKTDC
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Dynamic Bonds
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